U0126 | MEK選擇性非競爭型抑制劑 | 貨號1668-5 A MEK inhibitor Abcam操作手冊 (Abcam ab120241)
Alternate Name/Synonyms: 1,4-Diamino-2,3-dicyano-1,4-bis(o-aminophenylmercapto) butadiene
MAP kinase kinase(MEK)選擇性非競爭型抑制劑. Potent and selective non-competitive inhibitor of MAP kinase kinase(MEK). Inhibits MEK-1 and MEK-2 (IC₅₀ values of 0.07 and 0.06 µM respectively) with little or no effect on the activities of PKC, Abl, Raf, MEKK, ERK, JNK, MKK-3, MKK-4/SEK, MKK-6, Cdk2 or Cdk4. 分子型式C₁₈H₁₆N₆S₂ | 分子量Molecular Weight: 380.48 | 純度Purity: ≥98% by HPLC | Solubility: DMSO (>10 mg/ml)
Catalog # | Product Name+ | Size |
1594-100 | BAY 43-9006 | 100 mg |
1594-25 | BAY 43-9006 | 25 mg |
1954-5 | Doramapimod | 5 mg |
1954-25 | Doramapimod | 25 mg |
1783-5 | EZSolution™ PD 98059 | 5 mg |
1871-1 | EZSolution™ PD184352 | 1 mg |
1786-1 | EZSolution™ SB 203580 | 1 mg |
2729-5 | JNK-IN-8 | 5 mg |
2729-25 | JNK-IN-8 | 25 mg |
7011-50 | L-JNK Peptide Inhibitor I | 50 µl |
K862-7 | PathwayReady™ MAP Kinase Signaling Inhibitor Panel | 7 inhibitors |
1666-5 | PD 98059 | 5 mg |
1643-2 | PD-0325901 | 2 mg |
1643-5 | PD-0325901 | 5 mg |
1643-25 | PD-0325901 | 25 mg |
1585-25 | PD184352 | 25 mg |
1585-5 | PD184352 | 5 mg |
1585-1 | PD184352 | 1 mg |
1712-1 | SB 203580 | 1 mg |
1712-5 | SB 203580 | 5 mg |
1669-5 | SP600125 | 5 mg |
1668-5 | U0126 | 5 mg |
1598-1 | VX-702 | 1 mg |
1598-5 | VX-702 | 5 mg |
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